BDBM50391044 CHEMBL2088410

SMILES CC(=O)NCc1nc2cc(NC(=O)c3ccc(cc3)C(C)(C)C)ccc2s1

InChI Key InChIKey=HITAUNLFJVIXEG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50391044   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50391044(CHEMBL2088410)Copy SMILESCopy InChI

Affinity DataIC50: 2.42E+3nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor assessed as inhibition of capsaicin-induced calcium uptake by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/8/2013
Entry Details Article
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