BDBM50391052 CHEMBL2088419

SMILES CC(C)Oc1ccc(C(=O)Nc2ccc3sc(CO)nc3c2)c(C)c1

InChI Key InChIKey=MECQGLMDNYLKGI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50391052   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50391052(CHEMBL2088419)Copy SMILESCopy InChI

Affinity DataIC50: 47nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor assessed as inhibition of capsaicin-induced calcium uptake by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/8/2013
Entry Details Article
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