BDBM50393113 CHEMBL2153265

SMILES Nc1nc2c(nccc2[nH]1)-c1cccnc1

InChI Key InChIKey=CRSRGBLNXLTDTJ-UHFFFAOYSA-N

Data  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50393113   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Macquarie University

Curated by ChEMBL

LigandBDBM50393113(CHEMBL2153265)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using [gamma-32P] ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
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TargetCyclin-dependent kinase 5 activator 1(Human)
Macquarie University

Curated by ChEMBL

LigandBDBM50393113(CHEMBL2153265)Copy SMILESCopy InChI

Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-32P] ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL