BDBM50405897 CHEMBL5277241
SMILES CC(=O)OCc1ccc2sc(cc2c1)S(N)(=O)=O
InChI Key InChIKey=JPSSAXLGXLTVNR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50405897
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Incyte Research Institute
Curated by ChEMBL
Incyte Research Institute
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Incyte Research Institute
Curated by ChEMBL
Incyte Research Institute
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in guinea pig trachea in the presence of 11,9-epoxymethano-PGH2More data for this Ligand-Target Pair
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Incyte Research Institute
Curated by ChEMBL
Incyte Research Institute
Curated by ChEMBL
Affinity DataIC50: 409nMAssay Description:Inhibitory activity against Neisseria gonorrhoeae dihydrofolate reductase at 10e8 MMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibitory activity against Neisseria gonorrhoeae dihydrofolate reductase at 10e8 MMore data for this Ligand-Target Pair
Affinity DataIC50: 268nMAssay Description:Inhibitory activity against Neisseria gonorrhoeae dihydrofolate reductase at 10e8 MMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Affinity DataIC50: 198nMAssay Description:The compound was tested for alpha-adrenergic activity against Alpha-1 adrenergic receptor from rat aorta.More data for this Ligand-Target Pair