BDBM50413014 CHEMBL497171
SMILES CCCCNc1nccc2[nH]c3ccccc3c12
InChI Key InChIKey=IXKMSVHWGUFUOT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50413014
Affinity DataKi: 3.98nMAssay Description:Displacement of [125I]human urotensin 2 from human recombinant urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Displacement of [125I]human urotensin 2 from cat urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Antagonist activity at human urotensin 2 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of intercellular calcium mobilization ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.94nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair