BDBM50413567 CHEMBL511976

SMILES CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2c(F)c(F)c(F)c(F)c2F)CC1

InChI Key

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50413567   

TargetC-X-C chemokine receptor type 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413567(CHEMBL511976)
Affinity DataKi:  501nMAssay Description:Antagonist activity at human CXCR3 expressed in HEK293T cells coexpressing Galphaqi5 assessed as inhibition of CXCL10-induced [3H]inositol phosphate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413567(CHEMBL511976)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]CXCL10 from human CXCR3 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed