BDBM50433402 CHEMBL2380639

SMILES COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)c2ccccc12

InChI Key

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50433402   

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50433402(CHEMBL2380639)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50433402(CHEMBL2380639)
Affinity DataIC50: 36nMAssay Description:Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Rat)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50433402(CHEMBL2380639)
Affinity DataIC50: 70nMAssay Description:Inhibition of rat 11beta-HSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed