BDBM50444782 CHEMBL3099133
SMILES Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1ccccc1
InChI Key InChIKey=VRKJPABSKAXYBK-UHFFFAOYSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50444782
Affinity DataIC50: 85nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at CRTh2 in human RBC assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Antagonist activity at CRTh2 in human whole blood assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair