BDBM50448275 CHEMBL2414020

SMILES CCCOc1ccccc1-c1cc(no1)C(=O)NC12CC3CC(CC(C3)C1)C2

InChI Key

Data  2 KI  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50448275   

TargetCannabinoid receptor 2(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50448275(CHEMBL2414020)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO membranes assessed as [35S]-GTPgammaS binding after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50448275(CHEMBL2414020)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50448275(CHEMBL2414020)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50448275(CHEMBL2414020)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant FAAH expressed in Escherichia coli assessed as hydrolysis of [3H]-AEAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed