BDBM50456735 CHEMBL4204576
SMILES C[C@@H]1SC(=N[C@H]1Cc1c[nH]cn1)c1ccccc1
InChI Key InChIKey=OFXSSUCHCSBXFS-GWCFXTLKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50456735
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from human 5-HT7A receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University of The Philippines
Curated by ChEMBL
University of The Philippines
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at 5-HT7A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair