BDBM50473858 CHEMBL125758

SMILES [H][C@]12[C@@H](CC[C@@]1(CC[C@]1(C)[C@]2([H])CC[C@]2([H])[C@@]3(C)CC[C@H](O)C(C)(C)[C@]3([H])CC[C@@]12C)C(=O)NCc1ccc(O)c(OC)c1)C(C)=C

InChI Key InChIKey=VYRNPTYLGKJDHQ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50473858   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Istituto Per La Chimica Di Molecole Di Interesse Biologico

Curated by ChEMBL
LigandPNGBDBM50473858(CHEMBL125758)
Affinity DataEC50:  126nMAssay Description:Concentration necessary to induce a relative half-maximal response measured by the entry of [Ca2+] into human embryonic kidney HEK293 cells overexpre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed