BDBM50511176 CHEMBL4547545

SMILES CC1N(C(=O)NC1=O)c1cc(C)c(CCS(=O)(=O)N2CCC3(CC2)N=C(NC3=O)c2ccc(OC(F)(F)F)cc2)c(C)c1

InChI Key InChIKey=YPAKMWKBBYLLMB-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50511176   

TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Chugai Pharmaceutical

Curated by ChEMBL

LigandBDBM50511176(CHEMBL4547545)Copy SMILESCopy InChI

Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at recombinant human PTHR1 expressed in pig LLC-PK1 cells assessed as increase in cAMP production measured after 20 mins by EIAMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/20/2021
Entry Details Article
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