BDBM50512052 CHEMBL4446136
SMILES COc1ccccc1\C=C\C(=O)Nc1ccccc1C(O)=O
InChI Key InChIKey=YAYQPACFPAHFBP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50512052
TargetTransient receptor potential cation channel subfamily M member 8(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 5.01E+4nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as inhibition of CA-induced increase in calcium influx incubated for 10 mins pr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as inhibition of CA-induced increase in calcium influx incubated for 10 mins pr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataEC50: 7.50E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataEC50: 7.94E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair