BDBM50521198 CHEMBL4533807

SMILES [H][C@@]12C[C@@H](C)C[C@@]3([H])C(=O)\C(=C/NCCO)C(=O)[C@@](C)([C@@H](\C(C)=C\C)C(C)=C1)[C@]23[H]

InChI Key InChIKey=KXMSGRJOTFHUTA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521198   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
University of Utah

Curated by ChEMBL

LigandBDBM50521198(CHEMBL4533807)Copy SMILESCopy InChI

Affinity DataIC50: 6.16E+4nMAssay Description:Antagonist activity at human TRPM8 channel expressed in HEK293 cells assessed as inhibition of icilin-induced calcium flux by Fluo-4-AM dye based flu...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
Entry Details Article
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