BDBM50521887 CHEMBL4459939

SMILES C[C@H]1Cn2c(nc3ccccc23)N1C(=O)Cc1nc2c(C)ncc(C)n2n1

InChI Key InChIKey=AARRAQHMWVXNTL-LBPRGKRZSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521887   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50521887(CHEMBL4459939)Copy SMILESCopy InChI

Affinity DataIC50:  8.40nMAssay Description:Inhibition of human PDE10A using cAMP as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by HTRF detecti...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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