BDBM50528927 CHEMBL4517296
SMILES Cn1c(ccc1-c1cccc(OC(=O)NCCN2CCN(CC2)c2ccccc2)c1)C(N)=O
InChI Key InChIKey=JRYNLQPPXGHRTN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50528927
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 203nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 791nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataIC50: 6.46E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair