BDBM50528933 CHEMBL4449756

SMILES Cc1cc(C(N)=O)c(-c2cccc(OC(=O)NCCN3CCN(c4ccccc4)CC3)c2)[nH]1

InChI Key InChIKey=QZUKFTRCZFYKET-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50528933   

TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50528933BDBM50528933(CHEMBL4449756)
Affinity DataKi:  50nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50528933BDBM50528933(CHEMBL4449756)
Affinity DataIC50: 195nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed