BDBM50542765 CHEMBL4638592

SMILES CCP(=O)(OC)c1ccc2oc(nc2c1)-c1ccc(F)cc1

InChI Key InChIKey=MNCZMYLRBLYUPR-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50542765   

TargetUtrophin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  244nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  244nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  244nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  9.30E+3nMAssay Description:Antagonist activity at human Gq-coupled 5HT2B receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced calcium mobilization by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  9.30E+3nMAssay Description:Antagonist activity at human Gq-coupled 5HT2B receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced calcium mobilization by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50542765(CHEMBL4638592)
Affinity DataEC50:  711nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed