BDBM50552409 CHEMBL4785621

SMILES COc1ncccc1C(=O)N([C@@H](C(N)=O)c1ccccc1)[C@@H]1CCc2c1cc(Cl)cc2F

InChI Key InChIKey=YEGJBUBKJSSWNZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50552409   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Kissei Pharmaceutical

Curated by ChEMBL

LigandBDBM50552409(CHEMBL4785621)Copy SMILESCopy InChI

Affinity DataIC50: 380nMAssay Description:Antagonist activity at human TRPM8 transfected in HEK293T cells assessed as reduction in menthol-induced calcium influx measured after 60 mins by Flu...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/24/2022
Entry Details Article
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