BDBM50553839 CHEMBL4778103

SMILES FC(F)(F)c1cc(CNC(=O)Nc2cccc3[nH]ncc23)n(n1)-c1cccc(c1)C(F)(F)F

InChI Key InChIKey=XCWNXECPZLSFGJ-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50553839   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50553839(CHEMBL4778103)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO-K1 cells assessed as inhibition of capsaicin-induced Ca2+ response treated with compound 6 mins p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed