BDBM50566890 CHEMBL4865432
SMILES Fc1cnc(NCc2ccc(CNC(=O)c3ccc4nncn4c3)cc2)nc1
InChI Key InChIKey=JZMQONSLCVIHLI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50566890
Affinity DataIC50: 85nMAssay Description:Inhibition of human His-ENL YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity to human His-ENL YEATS domain assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >5.40E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 729nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair