BDBM50567081 CHEMBL4872408

SMILES CN(C)c1nccc(n1)-c1cnc2ncccn12

InChI Key InChIKey=UYXOVPJCCPREHU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50567081   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Sussex

Curated by ChEMBL

LigandBDBM50567081(CHEMBL4872408)Copy SMILESCopy InChI

Affinity DataIC50: 158nMAssay Description:Displacement of Kinase tracer 236 from biotinylated DYRK1A (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1.5 hrs by TR-FRET...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/19/2022
Entry Details Article
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