BDBM50583773 CHEMBL5091013

SMILES N=C(N)NCCC[C@@H](NC(=O)C=C(c1ccccc1)c1ccccc1)C(=O)NCC(N)=O

InChI Key InChIKey=ROWINWHJODIZTO-UHFFFAOYSA-N

Data  8 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50583773   

TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi:  1.69E+3nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF2 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Mouse)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [125I]-1DMeNPFF from mouse NPFF2R receptor by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPyroglutamylated RF-amide peptide receptor(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-Diprenorphine from human DOP receptor expressed in HEK293 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetProlactin-releasing peptide(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-PrRP-20 from human PrRP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in HEK293 cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Strasbourg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583773BDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]-Kp-10 from human Kiss1 receptor by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed