BDBM50592249 CHEMBL5191395
SMILES COc1ccc2sc(cc2c1)C(=O)N(C)Cc1cc(F)cc(F)c1
InChI Key InChIKey=FLWYCOJREJRWLJ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50592249
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant GST-tagged Clk1 (129 to 484 residues) expressed in Escherichia coli expression system using GRSRSRSRSRSRSRSR peptide ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
German University In Cairo
Curated by ChEMBL
German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Inhibition of human recombinant GST tagged full length DYRK1A expressed in Baculovirus expression system using GRSRSRSRSRSRSRSR peptide as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Inhibition of human recombinant GST-tagged Clk2 expressed in Baculovirus expression system using GRSRSRSRSRSRSRSR peptide as substrate in presence of...More data for this Ligand-Target Pair