BDBM50593386 CHEMBL5207050

SMILES Cc1cc(NC(=O)COc2ccc(C)cc2C)n(n1)C1CCS(=O)(=O)C1

InChI Key InChIKey=HGUSMXUDDLWABL-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50593386   

TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593386(CHEMBL5207050)
Affinity DataEC50:  1.74E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593386(CHEMBL5207050)
Affinity DataEC50:  5.54E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed