BDBM50600272 CHEMBL5204270
SMILES CN1CCC(CC1)c1ccc(cc1)-c1ccc2c(c1)ncn(C(C(=O)Nc1nccs1)c1ccccc1)c2=O
InChI Key InChIKey=KSCGLUWNVKAXQS-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50600272
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Dana-Farber Cancer Institute
Curated by ChEMBL
Dana-Farber Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibition of his-GST tagged human EGFR L858R/T790M double mutant expressed in insect cells incubated for 30 mins in presence of ATP by HTRF kinase a...More data for this Ligand-Target Pair