BDBM50600506 CHEMBL5203368

SMILES NC(=O)c1cc2c(cccc2s1)-c1ccc(s1)C(=O)NC1CC1

InChI Key InChIKey=QYQDTYWXMRWCEU-UHFFFAOYSA-N

Data  2 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50600506   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Ach£

Curated by ChEMBL

LigandBDBM50600506(CHEMBL5203368)Copy SMILESCopy InChI

Affinity DataKi:  160nMAssay Description:Inhibition of human DYRK1A incubated for 90 mins in presence of ATP by Z-LYTE based FRET assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/23/2023
Entry Details
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TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Ach£

Curated by ChEMBL

LigandBDBM50600506(CHEMBL5203368)Copy SMILESCopy InChI

Affinity DataKi:  670nMAssay Description:Inhibition of human DYRK1B incubated for 130 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/23/2023
Entry Details
Copy BDB DOIPubMed
Copy reaction URL