BDBM50606132 CHEMBL5197828

SMILES C[C@H](Oc1ccc(-c2nc3c(ncnc3[nH]2)C2=CCNCC2)c(F)c1)c1ccccc1

InChI Key InChIKey=GKWQGBRAJHDHPX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50606132   

TargetProtein arginine N-methyltransferase 5(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50606132(CHEMBL5197828)
Affinity DataIC50: 80nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed