BDBM50611362 CHEMBL5276538

SMILES CC(C)(C)n1nc(-c2ccc(NC(=O)c3cc(ccc3F)C(F)(F)F)cc2)c2c(N)ncnc12

InChI Key InChIKey=QBWCBCCHHYJEEW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50611362   

TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Yangtze University

Curated by ChEMBL
LigandPNGBDBM50611362(CHEMBL5276538)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant GST-tagged RET (unknown origin) using EAIYAAPFKKK as substrate in the presence of ATP of 100 uM by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed