BDBM50617291 CHEMBL5417678

SMILES CN(c1ncccc1CNc1ccnc(n1)-c1nc2ccc(cc2[nH]1)C#N)S(C)(=O)=O

InChI Key InChIKey=NLVVTXFNPRNRRC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50617291   

TargetSRSF protein kinase 1(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617291(CHEMBL5417678)
Affinity DataIC50: 324nMAssay Description:Inhibition of human SRPK1 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617291(CHEMBL5417678)
Affinity DataIC50: 3.77E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed