BDBM50635508 CHEMBL5527848

SMILES CC(C)c1cnn2c(NCc3ccc(NC(=O)C4(F)CC4)cc3)nc(NC3CCOCC3)nc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50635508   

TargetCyclin-dependent kinase 9(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50635508(CHEMBL5527848)
Affinity DataIC50: 28nMAssay Description:Inhibition of CDK9 (unknown origin) using ULight 4EBP1 peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 7(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50635508(CHEMBL5527848)
Affinity DataIC50: 261nMAssay Description:Inhibition of CDK7 (unknown origin) using ULight 4EBP1 peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50635508(CHEMBL5527848)
Affinity DataIC50: 806nMAssay Description:Inhibition of CDK2 (unknown origin) using ULight 4EBP1 peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50635508(CHEMBL5527848)
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of CDK4 (unknown origin) using ULight 4EBP1 peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 6(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50635508(CHEMBL5527848)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK6 (unknown origin) using ULight 4EBP1 peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed