BDBM50638593 CHEMBL5555026

SMILES CCC1(CC)CC(NC(=O)Nc2cccc3c(C)nccc23)c2cc(F)ccc2O1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50638593   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Hospital of Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50638593(CHEMBL5555026)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of NADA-induced increase in intracellular Ca2+ level incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Hospital of Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50638593(CHEMBL5555026)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed