BDBM50640172 CHEMBL5567647

SMILES CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)c1cc(C)cc(C)c1)C1CCCC1)C(=O)NCC(=O)N[C@H]1CCC(=O)OB1O

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50640172   

TargetSubtilisin-like protease 1(malaria parasite P. falciparum)
The Francis Crick Institute

Curated by ChEMBL
LigandPNGBDBM50640172(CHEMBL5567647)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
The Francis Crick Institute

Curated by ChEMBL
LigandPNGBDBM50640172(CHEMBL5567647)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed