BDBM50640314 CHEMBL5573333

SMILES CC(=O)C(=O)Nc1c(C)[nH]c(/C=C2\C(=O)Nc3ccc(C(=O)N[C@H](C)c4ccc(F)cc4)cc32)c1C

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50640314   

TargetG protein-coupled receptor kinase 5(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50640314(CHEMBL5573333)
Affinity DataIC50: 30nMAssay Description:Inhibition of human GRK5 (1 to 590) expressed in Escherichia coli using tubulin as substrate incubated for 5 mins in presence of [gamma-32P]-ATP by r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBeta-adrenergic receptor kinase 1(Bovine)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50640314(CHEMBL5573333)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of bovine GRK2 expressed in baculovirus infected insect cell using tubulin as substrate incubated for 5 mins in presence of [gamma-32P]-AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed