BDBM50642809 US20250195508, Name TL5-135

SMILES CCN1CCN(Cc2ccc(NC(=O)c3cc(Cl)cc(NC(=O)c4cncc(-c5cccs5)c4)c3)cc2C(F)(F)F)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50642809   

TargetEphrin type-A receptor 2(Human)
University of Central Florida Research Foundation

US Patent
LigandPNGBDBM50642809(US20250195508, Name TL5-135)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro biochemical kinase assays were done using recombinant human EPHA2. compounds were subjected to in vitro biochemical kinase assays done using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

TargetEphrin type-A receptor 2(Human)
University of Central Florida Research Foundation

US Patent
LigandPNGBDBM50642809(US20250195508, Name TL5-135)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EphA2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed