BDBM50647168 CHEMBL5596085

SMILES CC(C)(C)OC(=O)N1CCN(Cc2ccc3nc(NC(=O)c4ccc(S(=O)(=O)NCCC#N)cc4)sc3c2)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50647168   

TargetProprotein convertase subtilisin/kexin type 9(Human)
Hebei Normal University

Curated by ChEMBL
LigandPNGBDBM50647168(CHEMBL5596085)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of PCSK9 transcriptional activity in human HepG2 cells by luciferase reporter based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed