BDBM50652127 CHEMBL5647058

SMILES COc1c(N2C[C@@H]3CCCN(Cc4cnc(C)c(O)c4C)[C@@H]3C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50652127   

TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Kazan (Volga region) Federal University

Curated by ChEMBL
LigandPNGBDBM50652127(CHEMBL5647058)
Affinity DataIC50: 16nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase-IV assessed as reduction in decatenation using kinetoplast DNA as substrate incubated for 30 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Kazan (Volga region) Federal University

Curated by ChEMBL
LigandPNGBDBM50652127(CHEMBL5647058)
Affinity DataIC50: 52nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using relaxed pBR322 DNA as substrate incubated for 30 mins by ethidium bromide staining based agarose...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Kazan (Volga region) Federal University

Curated by ChEMBL
LigandPNGBDBM50652127(CHEMBL5647058)
Affinity DataIC50: 400nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using supercoiled pBR322 DNA as substrate incubated for 60 mins by ethidium bromide staining based aga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed