BDBM509688 4-[[2-(5-Chloro-2-hydroxy-phenyl)acetyl]amino]-N-(4-cyanotetrahydropyran-4-yl)pyridine-2-carboxamide::US11364246, Example 31::US20200361871A1, Example 31
SMILES Oc1ccc(Cl)cc1CC(=O)Nc1ccnc(c1)C(=O)NC1(CCOCC1)C#N
InChI Key InChIKey=QXLCCQLDHASOPP-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 509688
Affinity DataEC50: 120nMAssay Description:Cell Culture and PreparationFisher rat thyroid (FRT) cells stably expressing human TMEM16A (TMEM16Aabc variant; Dr Luis Galietta, Insituto Giannina, ...More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair