BDBM513779 US11091495, Example 140

SMILES Fc1ccc2OCCc2c1CNc1ncc(N2CCNCC2)c2nc(cn12)C#N

InChI Key InChIKey=HPRRNWSWKSVYEO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 513779   

TargetHistone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2(Human)
Mirati Therapeutics

US Patent

LigandBDBM513779(US11091495, Example 140)Copy SMILESCopy InChI

Affinity DataIC50: 500nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
1/30/2022
Entry Details
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