BDBM5212 2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-5- ((4-methylpyrimidin-5-yl)oxy)-1H-indazol- 4-yl)amino)isoindoline-1,3-dione::US20240208937, Compound 26

SMILES Cc1ncncc1Oc1ccc2c(cnn2C)c1Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O

InChI Key InChIKey=OHDFAXVXAMAICU-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 5212   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5212BDBM5212(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-5- ((4-me...)
Affinity DataEC50:  55nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5212BDBM5212(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-5- ((4-me...)
Affinity DataEC50: >100nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent