BDBM524270 Preparation of Ethyl 5-methyl-1-((2-(piperidin-1-yl)thiazol-4-yl)methyl)-1H-pyrrole-2-carboxylate::US11168080, Compound A-39::US11168080, Compound A-42

SMILES Cc1ccc(C(=O)Nc2ccccc2)n1Cc1csc(n1)N1CCCCC1

InChI Key InChIKey=IHZIPLLKNYVYIO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 524270   

TargetDynamin-1-like protein(Human)
Mitobridge

US Patent
LigandPNGBDBM524270(US11168080, Compound A-39 | US11168080, Compound A...)
Affinity DataIC50: 2.60E+4nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetDynamin-1-like protein(Human)
Mitobridge

US Patent
LigandPNGBDBM524270(US11168080, Compound A-39 | US11168080, Compound A...)
Affinity DataIC50: 3.60E+4nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent