BDBM524297 Preparation of 4-(4-bromo-1-((2-(piperidin-1-yl)thiazol-4-yl)methyl)-1H-pyrrole-2-carboxamido)benzoic Acid::US11168080, Compound A-64

SMILES OC(=O)c1ccc(NC(=O)c2cc(Br)cn2Cc2csc(n2)N2CCCCC2)cc1

InChI Key InChIKey=VSOLWKUTROLZEM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 524297   

TargetDynamin-1-like protein(Human)
Mitobridge

US Patent
LigandPNGBDBM524297(Preparation of 4-(4-bromo-1-((2-(piperidin-1-yl)th...)
Affinity DataIC50: 1.00E+5nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent