BDBM5276 4-((6-(2,3-dimethylpyridin-4-yl)-1-methyl- 1H-indazol-5-yl)amino)-2-(2,6- dioxopiperidin-3-yl)isoindoline-1,3-dione::US20240208937, Compound 29

SMILES Cc1nccc(-c2cc3c(cnn3C)cc2Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1C

InChI Key InChIKey=WORFIAYAIJPLPO-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 5276   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5276BDBM5276(4-((6-(2,3-dimethylpyridin-4-yl)-1-methyl- 1H-inda...)
Affinity DataEC50:  55nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5276BDBM5276(4-((6-(2,3-dimethylpyridin-4-yl)-1-methyl- 1H-inda...)
Affinity DataEC50: >100nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent