BDBM529371 US11198699, Compound 1
SMILES C[C@]1(CCc2ccc3cc(Br)c(N)nc3c2)C[C@H]([C@H](O)[C@@H]1O)n1ccc2c(N)ncnc12
InChI Key InChIKey=TYWVDVASSSOQLE-XQQXVUDOSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 529371
TargetMethylosome protein 50/Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Aligos Therapeutics
US Patent
Aligos Therapeutics
US Patent
Affinity DataIC50: <1nMAssay Description:Assay 2: Compounds were tested for inhibition of methyltransferase activity in 384-well plate assay format using mass spectrometry technology. In thi...More data for this Ligand-Target Pair
TargetMethylosome protein 50/Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Aligos Therapeutics
US Patent
Aligos Therapeutics
US Patent
Affinity DataIC50: <1nMAssay Description:Assay 1: Compounds were tested for inhibition of methyltransferase activity in a radioisotope filter binding assay, similar to previously described i...More data for this Ligand-Target Pair