BDBM530563 WO2022076495, EXAMPLE 9

SMILES CCOc1cccc(c1)-n1c2ccc(cc2n(C(C)C)c1=O)C(=O)NC1(C)CS(=O)(=O)C1

InChI Key InChIKey=QRAOXNRRCUABRE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 530563   

TargetDiacylglycerol O-acyltransferase 2(Human)
Merck Sharp &Amp

WIPO
LigandPNGBDBM530563(WO2022076495, EXAMPLE 9)
Affinity DataIC50:  4.30nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product 13Ci8-triolein (13C-l,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails WIPO WO2022076495