BDBM534169 N-(Benzenesulfonyl)-6-cyclopropyl-4-(dimethylamino)benzofuran-2-carboxamide::WO2022081842, Example 42

SMILES CN(C)c1cc(cc2oc(cc12)C(=O)NS(=O)(=O)c1ccccc1)C1CC1

InChI Key InChIKey=NWTHEADRPSSHGE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534169   

TargetHistone acetyltransferase KAT6A [507-778](Human)
The Broad Institute

WIPO
LigandChemical structure of BindingDB Monomer ID 534169BDBM534169(WO2022081842, Example 42 | N-(Benzenesulfonyl)-6-c...)
Affinity DataIC50: 417nMAssay Description: Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081842