BDBM5373 2-(2,6-dioxopiperidin-3-yl)-4-((6-methoxy- 4-phenylpyridin-3-yl)amino)isoindoline- 1,3-dione::US20240208937, Compound 30

SMILES COc1cc(-c2ccccc2)c(Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cn1

InChI Key InChIKey=ZEXKFKBEVSHKSG-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 5373   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5373BDBM5373(2-(2,6-dioxopiperidin-3-yl)-4-((6-methoxy- 4-pheny...)
Affinity DataEC50:  55nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 5373BDBM5373(2-(2,6-dioxopiperidin-3-yl)-4-((6-methoxy- 4-pheny...)
Affinity DataEC50:  55nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent