BDBM6284 2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (4-methylthiazol-2-yl)-2-oxo-1,2,3,4- tetrahydroquinolin-7-yl)amino)isoindoline- 1,3-dione::US20240208937, Compound 39

SMILES Cc1csc(-c2cc3c(cc2Nc2cccc4c2C(=O)N(C2CCC(=O)NC2=O)C4=O)N(C)C(=O)CC3)n1

InChI Key InChIKey=TUTFKQIOTHPXAR-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 6284   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 6284BDBM6284(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (4-met...)
Affinity DataEC50:  55nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 6284BDBM6284(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (4-met...)
Affinity DataEC50:  55nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent