BDBM660630 N-(6-chloropyridin-3-yl)-4- methoxy-1H-pyrrolo[2,3- c]pyridin-7-amine formate::US20240101531, Example 15

SMILES COc1cnc(Nc2ccc(Cl)nc2)c2[nH]ccc12

InChI Key InChIKey=IOUWWPAVUMTMJK-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 660630   

TargetPotassium voltage-gated channel subfamily KQT member 2/3 (Human)
Xenon Pharmaceuticals

US Patent
LigandPNGBDBM660630(N-(6-chloropyridin-3-yl)-4- methoxy-1H-pyrrolo[2,3...)
Affinity DataEC50:  5.50E+3nMAssay Description:This potassium flux assay employs the cell-permeable, potassium-sensitive dye, IPG-2 AM, to quantify potassium ion flux through potassium channels.In...More data for this Ligand-Target Pair
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Date in BDB:
6/11/2024
Entry Details
US Patent