BDBM685120 US12565480, Compound 2::US20240239763, Compound Formula I
SMILES OC(=O)c1ccc(cc1O)-c1sc(C#N)c2CCC(F)(F)Cc12
InChI Key InChIKey=UTTXOYFICPSQLS-UHFFFAOYSA-N
Data 13 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 685120
Affinity DataIC50: 20.7nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of XO (unknown origin) using xanthine as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of XO (unknown origin) using xanthine as substrate assessed as decrease in uric acid level by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+4nMAssay Description:Test compounds, standard inhibitors (at 100× final concentration), and mixed substrate working solutions were prepared; the microsomes (purchased fro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Test compounds, standard inhibitors (at 100× final concentration), and mixed substrate working solutions were prepared; the microsomes (purchased fro...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Test compounds, standard inhibitors (at 100× final concentration), and mixed substrate working solutions were prepared; the microsomes (purchased fro...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Test compounds, standard inhibitors (at 100× final concentration), and mixed substrate working solutions were prepared; the microsomes (purchased fro...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Test compounds, standard inhibitors (at 100× final concentration), and mixed substrate working solutions were prepared; the microsomes (purchased fro...More data for this Ligand-Target Pair